EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.3.2.13 | 0.0000021 |
- |
methyl 4-[[(bromoacetyl)oxy]methyl]benzoate |
at pH 7.1, temperature not specified in the publication |
735930 |
2.3.2.13 | 0.0000039 |
- |
2-bromo-1-(tricyclo[3.3.1.13,7]dec-1-yl)ethanone |
at pH 7.1, temperature not specified in the publication |
735930 |
2.3.2.13 | 0.0000061 |
- |
N-(2-[4-[5-(dimethylamino)naphthalene-1-sulfonyl]piperazin-1-yl]-2-oxoethyl)prop-2-enamide |
at pH 7.1, temperature not specified in the publication |
735930 |
2.3.2.13 | 0.00000629 |
- |
tricyclo[3.3.1.13,7]dec-1-ylmethyl bromoacetate |
at pH 7.1, temperature not specified in the publication |
735930 |
2.3.2.13 | 0.00000665 |
- |
methyl 6-[[(chloroacetyl)oxy]methyl]naphthalene-2-carboxylate |
at pH 7.1, temperature not specified in the publication |
735930 |
2.3.2.13 | 0.00000875 |
- |
2-chloro-1-(tricyclo[3.3.1.13,7]dec-1-yl)ethanone |
at pH 7.1, temperature not specified in the publication |
735930 |
2.3.2.13 | 0.00001 |
- |
N-[4-[4-(adamantane-1-carbonyl)piperazine-1-sulfonyl]-phenyl]acrylamide |
in 25 mM HEPES, pH 7.4, 250 mM NaCl, 2 mM MgCl2, 10 mM CaCl2, 0.2 mM dithiothreitol, and 0.05% (v/v) Pluronic F-127 at 37°C |
720194 |
2.3.2.13 | 0.000014 |
- |
N-[5-[4-(adamantane-1-carbonyl)piperazine-1-sulfonyl]-pyrimidin-2-yl]acrylamide |
in 25 mM HEPES, pH 7.4, 250 mM NaCl, 2 mM MgCl2, 10 mM CaCl2, 0.2 mM dithiothreitol, and 0.05% (v/v) Pluronic F-127 at 37°C |
720194 |
2.3.2.13 | 0.000015 |
- |
methyl 6-[[(bromoacetyl)oxy]methyl]naphthalene-2-carboxylate |
at pH 7.1, temperature not specified in the publication |
735930 |
2.3.2.13 | 0.000015 |
- |
N-[5-[4-(adamantane-1-carbonyl)piperazine-1-sulfonyl]-pyridin-2-yl]acrylamide |
in 25 mM HEPES, pH 7.4, 250 mM NaCl, 2 mM MgCl2, 10 mM CaCl2, 0.2 mM dithiothreitol, and 0.05% (v/v) Pluronic F-127 at 37°C |
720194 |