EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.8.1.7 | 0.00015 |
- |
5-hydroxy-1,4-naphthoquinone |
pH 7.0, 0.1 M potassium phosphate, 1 mM EDTA, 25°C |
711008 |
1.8.1.7 | 0.00033 |
- |
Hg2+ |
- |
394708 |
1.8.1.7 | 0.00035 |
- |
Cu+ |
pH 7.8, 37°C |
742059 |
1.8.1.7 | 0.0004 |
- |
5-(4-chlorophenyl)-8-fluoro-2-methyl-5a,9a-dihydropyrido[3,4-b]quinoxaline-1,3(2H,5H)-dione |
pH 6.9, 25°C |
659698 |
1.8.1.7 | 0.0005 |
- |
2,4,6-trinitrobenzene-sulfonate |
below, at 50% inhibition value, leading to oxidase activity |
394708 |
1.8.1.7 | 0.0005 |
- |
2-methyl-5-(1-naphthyl)-5a,9a-dihydropyrido[3,4-b]quinoxaline-1,3(2H,5H)-dione |
pH 6.9, 25°C |
659698 |
1.8.1.7 | 0.0006 |
- |
5,8-Dihydroxy-1,4-naphthoquinone |
pH 7.0, 0.1 M potassium phosphate, 1 mM EDTA, 25°C |
711008 |
1.8.1.7 | 0.0006 |
- |
5-(4-chlorophenyl)-5a,9a-dihydropyrido[3,4-b]quinoxaline-1,3(2H,5H)-dione |
pH 6.9, 25°C |
659698 |
1.8.1.7 | 0.0008 |
- |
ketotifen |
in 40 mM Tris-HCl buffer, pH 8.0, at 25°C |
725616 |
1.8.1.7 | 0.0008 |
- |
Zn2+ |
at 50% inhibition value |
394708 |